Tag: Binding affinity

Application of a macrocyclization strategy in kinase inhibitor development

Announcing a new publication for Acta Materia Medica journal. Kinases have a pivotal role in phosphorylation and kinase dysregulation has been implicated in the occurrence and progression of various diseases. By mid-2024 the Food and Drug Administration had approved 81 small-molecule kinase inhibitors targeting greater than 30 kinases, providing substantial clinical benefits for patients with […]